Anastrazolos 1 has an active substance Anastrozole. It is a popular inhibitor of aromatase and most recently appeared in the sports market. Initially, the drug was created to prevent breast cancer. The drug can reduce estrogen in the circulatory system and slow inflammation. Anastrazolos can be bought at an optimal price.
Basically, bodybuilders use the drug to eliminate the negative effects that appear due to the use of steroid drugs. The remedy is used by professional athletes on long courses of strong steroids. Anastrazolos, the price of which is acceptable for each athlete, gives excellent results in powerful cycles.
The drug has an active ingredient anastrozole. It is a selective inhibitor of aromatase, an enzyme involved in the process of aromatization, the formation of estrogen (female) hormones. Initially, anastrozole, like its analogues letrozole and vorozole, was developed and produced only for use in medicine: for tumors of the breast (breast) and other oncological diseases in women.
Anastrazolos 1(anastrozole) refers to the third, last generation of aromatase inhibitors. From antiestrogenic tamoxifen and clomiphene, citrate differs not only in the power of the effect, but in the mechanism of action (tamoxifen and clomiphene, according to the type of action, are blockers of estrogen receptors).
Anastrazolos 1 is not a steroid drug – it does not have pronounced anabolic, androgenic or progestagenic properties (but it can indirectly, by feedback, when a decrease in the level of estrogen leads to an increase in the level of androgens, promote anabolic and androgenic processes, reduce the fat layer and eliminate excess fluid).
Antiestrogen Anastrazolos rarely provokes side effects. But completely exclude the possibility of manifestations of violations from the central nervous, digestive, endocrine systems, as well as metabolism and allergic reactions can not. In order to exclude potential risks, it is recommended to be examined before reception, to get a specialist’s advice and, if necessary, to take tests, otherwise nothing guarantees harmlessness.
It is important that the reviews of Anastrazolos (1 mg / tab, 100 tab) are more often described as laudatory, as the antiestrogenic effect of the drug develops in a short time, and its own side effects are the exception to the rules (or the result of mistakes made during reception). The manufacturer of PharmaCom Labs has proven itself.
How to take Anastrazolos 1?
With the proper construction of the drug, the drug effectively treats and prevents the appearance of estrogenic side effects, such as excessive water retention, suppression of testosterone production, fat enlargement, gynecomastia and others. Therefore, it is relevant for use in sports practice.
The average recommended dose of Anastrazolos varies from 250 mg per day to 1 mg per day (the drug is not long-acting, so intensive use is necessary for optimal effect). Effective doses are selected individually, depending on the needs and tolerability of the body.
Reception Anastrazolosa can be carried out, at least, two schemes: 1st – to prevent estrogen-dependent side effects (from the first weeks of the course in the prophylactic dosage – an average of 0.5 mg every other day or every day); 2 nd – for treatment after symptoms of estrogenic side effects (symptomatically in a full dose – an average of 1 mg daily).
The course of taking Anastrazolos is not associated with an increased risk of its own side effect, but before exercise requires the elimination of contraindications. Among them: liver failure, kidney failure, childhood, pregnancy, breast-feeding, premenopause, hypersensitivity.
Effect and properties Anastrazolos 1
The active substance of this drug, anastrozole, was developed back in the 90s by Zeneca Pharmaceuticals, and at the end of 1995 it was approved for use in the United States. It was created exclusively for medical purposes as a new and effective means for the treatment of cancer, in particular for the treatment of operable breast cancer in women.At that time, anastrozole was the first such remedy in its class (that is, it was the first aromatase inhibitor of the third generation, among which today is also commonly referred to letrozole and vorozole)
If you describe specifically Anastrazolos 1 , then first of all it is worth noting that the mechanism of action of the drug is associated with the inhibition of aromatase in peripheral tissues, including fatty tissue. After intake, it is quickly absorbed from the gastrointestinal tract and also quickly takes up the case (Cmax in the blood, by the way, is reached already within the first few hours after administration). Food intake can slow the absorption rate somewhat, however, it does not affect the degree of absorption.
As a result, the effect of Anastrazolos 1 in tablets is rapid and powerful – the drug is able to effectively inhibit aromatase, as a consequence, blocking the process of aromatization, reducing and not allowing the level of estrogen to increase. This action is valuable not only when applied in medicine, but also important for athletes. In particular, it is highly regarded by athletes who use flavoring steroids that can lead to the development of estrogenic side effects, for example, to gynecomastia.
Anastrazolos 1 is excreted, as it exerts its effect, also quickly enough (most of the drug is excreted in the urine within 72 hours after a single application).
Can Anastrazolos 1 itself cause side effects? Some risks are present, in particular, such abnormalities as: nausea, vomiting, diarrhea, anorexia, weakness or drowsiness, hot flushes, or headaches may tell about yourself. There is a possibility of some other side effects, including allergic reactions, so the use of these tablets should be approached with all seriousness, without violating the recommendations.
At Storage conditions of tablets: after purchase, they should be stored in a place inaccessible to moisture and light. Storage temperature – usually room, without sudden changes, as they can damage efficiency.
Positive qualities and effects
- Suppresses aromatization;
- The level of testosterone rises;
- Has an inhibitory effect;
- There is no estrogenic activity;
- The drug is not a steroid;
- Half of estrogens are suppressed;
- Progestogens are not active.
Methods of application and dosage Anastrazolos 1
Anastrazolos 1 is used by professional athletes on long cycles of steroids with the risk of appearance of aromatization. It is not recommended to apply the drug to women, because they may have undesirable consequences.
There are several regimens for applying the Anastrazolos 1 course. The first scheme is that the tablets consume at the first signs of aromatization in a dose of 0.25-1 milligram each day. The second scheme is the use of the drug from the beginning of the course of steroids in small dosages to prevent negative reactions of the body.
It is best to use Anastrazolos tablets on an empty stomach, drinking plenty of water. So the drug is much more quickly absorbed in the body and does not disrupt the work of the stomach and intestines. Before the beginning of the course it is advisable to consult with a specialist.
Reviews about Anastrazolos 1
About Anastrazolos 1 athletes mostly respond positively. This drug helps athletes eliminate side effects on the cycle and normalize the body. The drug is quite effective and safe, provided that the recommended dosages are observed. Athletes say that if there are signs of aromatization or gynecomastia, immediately it is necessary to resort to the use of Anastrazolos 1. It is best to ask the doctor what dosages may suit you.